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Updated: May 24, 2025

Modification and Functionalization of the Guanidine Group by Tailor-made Precursors
09:45

Modification and Functionalization of the Guanidine Group by Tailor-made Precursors

Published on: April 27, 2017

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作为具有抗增殖活性的多功能血清激素受体配体的长链循环阿里尔瓜尼丁

Przemysław Zaręba1, Anna K Drabczyk2, Artur Wnorowski3

  • 1Faculty of Chemical Engineering and Technology, Department of Chemical Technology and Environmental Analytics, Cracow University of Technology, 24 Warszawska Street, 31-155 Cracow, Poland.

ACS omega
|March 3, 2025
PubMed
概括

针对5-HT6R的新型多功能血清素受体配体显示出针对质瘤细胞的显著抗癌活性. 这些新型化合物显示出对癌症治疗的潜力,特定的配体显示出高疗效.

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Functionalized Spirocyclic Heterocycle Synthesis and Cytotoxicity Assay

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