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Updated: May 24, 2025

Monitoring GPCR-β-arrestin1/2 Interactions in Real Time Living Systems to Accelerate Drug Discovery
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Published on: June 28, 2019

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发现GPCR药物:新的药物,标和适应症

Javier Sánchez Lorente1, Aleksandr V Sokolov2, Gavin Ferguson1,3

  • 1Department of Drug Design and Pharmacology, Faculty of Health and Medical Sciences, University of Copenhagen, Copenhagen, Denmark.

Nature reviews. Drug discovery
|March 3, 2025
PubMed
概括

G蛋白结合受体 (GPCR) 是主要的药物标,有516种已批准的药物和337种正在临床试验中. 研究表明,在代谢性疾病,瘤学和免疫学中,GPCR药物开发的增加.

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