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Updated: May 24, 2025

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虚拟库对接可用于具有减少副作用的大麻素-1受体激动剂.

Tia A Tummino1,2, Christos Iliopoulos-Tsoutsouvas3, Joao M Braz4

  • 1Department of Pharmaceutical Chemistry, University of California, San Francisco, San Francisco, CA, 94158, USA.

Nature communications
|March 5, 2025
PubMed
概括

研究人员发现了新的大麻素化学型,它们作为大麻素-1受体 (CB1R) 的激动剂. 这些化合物显示出缓解疼痛的潜力,将止痛作用与常见的大麻素副作用分开.

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