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Updated: May 20, 2025

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克莱博普里德可以刺激人类心房中的5-HT4-色素受体

Lina Maria Rayo Abella1, Joachim Neumann2, Britt Hofmann3

  • 1Medical Faculty, Institute for Pharmacology and Toxicology, Martin Luther University Halle-Wittenberg, Magdeburger Straße 4, D-06112, Halle (Saale), Germany.

Naunyn-Schmiedeberg's archives of pharmacology
|March 25, 2025
PubMed
概括

克莱博普里德在人类心脏5-HT4血清素受体中充当激动剂和对抗剂. 这种药物增强了心脏收缩,特别是与西洛斯塔米德 (cilostamide) 结合时,它还可以抑制血清素诱导的效应.

关键词:
5HT4 - 血清素受体的受体克莱博普里德 (Clebopride) 是一种药物.人类心房是人的心房.转基因小鼠的研究结果

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