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Updated: May 20, 2025

Preparation and Characterization of Lipophilic Doxorubicin Pro-drug Micelles
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作为一种提高药物透性的策略,亲药方法

Mateus Mello de Souza1, Ana Luísa Rodriguez Gini1, Jhonnathan Alves Moura2

  • 1School of Pharmaceutical Sciences, São Paulo State University (UNESP), Araraquara 14800-903, SP, Brazil.

Pharmaceuticals (Basel, Switzerland)
|March 27, 2025
PubMed
概括

前药物增强药物的吸收和透性,这对于有效的药物输送至关重要. 本综述探讨了前药物策略,包括在PROteolysis TTargeting Chimeras (PROTACs) 中的应用,以提高药物的有效性和安全性.

关键词:
这就是PROTAC.发现药物的发现.药物的透性 药物的透性分子优化分子优化透性 透性的药物前体是药物前体.

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