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Updated: May 5, 2026

Preparation of Stable Bicyclic Aziridinium Ions and Their Ring-Opening for the Synthesis of Azaheterocycles
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Preparation of Stable Bicyclic Aziridinium Ions and Their Ring-Opening for the Synthesis of Azaheterocycles

Published on: August 22, 2018

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通过 [3+2] - 循环添加的Spiro[1-azabicyclo[3.2.0]heptane]框架的高效合成

Yulia Pronina1, Alexander Filatov1, Stanislav Shmakov2

  • 1Saint Petersburg State Institute of Technology, Moskovskii pr. 26, St. Petersburg 190013, Russian Federation.

The Journal of organic chemistry
|March 27, 2025
PubMed
概括

这项研究引入了一种高效的单合成新型聚环化合物使用亚甲化物. 该方法产生具有高立体选择性的螺旋和离散结构,显示出新药发现的潜力.

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