相关实验视频

Updated: Jul 14, 2026

Preparation of N-(2-alkoxyvinyl)sulfonamides from N-tosyl-1,2,3-triazoles and Subsequent Conversion to Substituted Phthalans and Phenethylamines
10:42

Preparation of N-(2-alkoxyvinyl)sulfonamides from N-tosyl-1,2,3-triazoles and Subsequent Conversion to Substituted Phthalans and Phenethylamines

Published on: January 3, 2018

用1,3,4-oxadiazole重新定位甲醇支架,以获得选择性,强效和耐受良好的抗真菌活性

Mohamed Hagras1, Hany G Ezzat1, Abdelrahman A Abuelkhir1

  • 1Department of Pharmaceutical Organic Chemistry, College of Pharmacy, Al-Azhar University Cairo 11884 Egypt m.hagrs@azhar.edu.eg.

RSC advances
|March 28, 2025
PubMed
概括

新型基于菲尼尔亚zole的oxadiazole衍生品显示强大的抗真菌活性对抗耐药菌株,如Candida auris. 化合物35是一种有前途的领先候选物,具有良好的安全性,解决了迫切需要新的抗真菌疗法.

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