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Updated: May 16, 2025

A High-Throughput Luciferase Assay to Evaluate Proteolysis of the Single-Turnover Protease PCSK9
08:14

A High-Throughput Luciferase Assay to Evaluate Proteolysis of the Single-Turnover Protease PCSK9

Published on: August 28, 2018

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用于治疗高胆固醇血症的口服PCSK9抑制剂:PURSUIT随机试验

Michael J Koren1, Rick B Vega2, Nikhil Agrawal3

  • 1Jacksonville Center for Clinical Research, Flourish Research Group, Jacksonville, Florida, USA.

Journal of the American College of Cardiology
|April 1, 2025
PubMed
概括

AZD0780,是一种口服的プロ蛋白转化酶亚素/素9型 (PCSK9) 抑制剂,在高胆固醇血症患者中显著降低了LDL-C. 这种新型治疗方法显示出良好的安全性,支持其进一步开发用于日常使用.

关键词:
在ACC/AHA的指导方针中.AZD078080 在线观看这就是LDL-C.抑制PCSK9的发生.超高胆固醇血症是一种高胆固醇血症.

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