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Updated: May 17, 2025

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硫素启发的N-phosphonopiperidones作为选择性的共价DPP8和DPP9抑制剂

Leonard Sewald1, Werner W A Tabak1, Lorenz Fehr1

  • 1Chemical Biology, Center of Medical Biotechnology, Faculty of Biology, University Duisburg-Essen, Essen, Germany.

Nature communications
|April 3, 2025
PubMed
概括

研究人员开发了针对二二酶 (DPP) 8和9 (DPP8 / 9) 的新型共价抑制剂. 微调化学弹头的微调.

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