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Updated: May 15, 2025

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对于Mu阿片类受体偏向激素的预测模型

Fernando J Tun-Rosado1, Elier E Abreu-Martínez2, Axel Magdaleno-Rodriguez1

  • 1Instituto de Química, Unidad Mérida, Universidad Nacional Autónoma de México, Carretera Mérida-Tetiz Km. 4.5, Ucú, Yucatán 97357, México.

Biochemistry
|April 10, 2025
PubMed
概括

开发更安全的阿片类药物疗法需要理解mu-opioid受体 (MOR) 偏倚的激素. 这项研究分析了偏向的MOR激动剂,揭示了更安全的药物设计的关键分子特征和相互作用.

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