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Updated: May 17, 2025

A Method for Screening and Validation of Resistant Mutations Against Kinase Inhibitors
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新的激酶抑制剂对瘤细胞具有选择性细胞毒性

D A Skvortsov1, I V Zhirkina2, D A Ipatova2

  • 1Chemistry Department and Belozersky Institute of Physico-Chemical Biology, Moscow State University, Moscow, Russia. skvorratd@mail.ru.

Doklady. Biochemistry and biophysics
|April 11, 2025
PubMed
概括

研究人员发现了新的多酶抑制剂STOCK7S-36520和STOCK7S-47016,它们可以选择性地向瘤细胞. 这些化合物通过抑制特定的激酶,如GCK.这些化合物显示出癌症治疗的希望.

关键词:
在FCCT的测试试验中.抗癌药物 抗癌药物 抗癌药物细胞毒性 细胞毒性激酶抑制剂 激酶抑制剂选择性的选择性

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