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Updated: May 13, 2025

A Novel In vitro Model for Studying the Interactions Between Human Whole Blood and Endothelium
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人类前环和血栓素合成酶:分子相互作用,调节和药理学

Pavel V Ershov1, Evgeniy O Yablokov1, Yuri V Mezentsev1

  • 1Institute of Biomedical Chemistry, 10, Pogodinskaya Street, 119121, Moscow, Russia.

Biochimie
|April 13, 2025
PubMed
概括

本综述检查了前环素合成酶 (PTGIS) 和血栓素合成酶 (TBXAS1),这是前列腺路中的关键酶. 了解它们的调节为心血管疾病和癌症提供了洞察力,TBXAS1抑制剂显示出更有前临床前景.

关键词:
药物发现 药物发现在PTGIS中使用.在临床前的药理学.простациклин合成酶 的使用方法蛋白质与蛋白质的相互作用这就是TBXAS1的原因.血素合成酶的使用方法

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