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Updated: May 13, 2025

Microwave-Assisted Preparation of 1-Aryl-1H-pyrazole-5-amines
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合成,生物活性和分子对接研究:新型arylpiperazine衍生物作为潜在的新耐药AR抗剂

Hua Jiang1, Haowei Chen2, Ya Wang2

  • 1Department of Urology, The Fifth Affiliated Hospital of Zunyi Medical University (Zhuhai Sixth People's Hospital), Zhuhai, China.

Frontiers in chemistry
|April 14, 2025
PubMed
概括

研究人员发现了作为雄激素受体对抗剂的新化合物,显示了治疗荷尔蒙抵抗性前列腺癌 (PCa) 的潜力. 这些新型药物有效地减少了癌细胞的生长,并向了雄激素受体通路.

关键词:
抗逆转基因抗生素对手具有对抗性的活动.结合的亲和关系是有约束力的.停靠研究对接研究前列腺癌是前列腺癌.

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