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Updated: May 13, 2025

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6 - 亚里尔异印-1-单元:新型mGluR2 负基调节剂

Yinlong Li1, Steven H Liang1

  • 1Department of Radiology and Imaging Sciences, Emory University, 1364 Clifton Road, Atlanta, Georgia 30322, United State.

ACS medicinal chemistry letters
|April 16, 2025
PubMed
概括

研究人员开发了新的化合物,即6 - 烯异印-1-衍生物,它们对甲基酸盐受体2 (mGluR2) 起负基调制剂 (NAM) 的作用. 这项研究详细介绍了它们的合成,并评估了它们对mGluR2和mGluR3.3的功效.

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