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Updated: May 11, 2025

Spectrophotometric Screening for Potential Inhibitors of Cytosolic Glutathione S-Transferases
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新型非类固醇类固醇硫酶抑制剂含有谷氨酸单元的谷氨酸酸

Olga Ciupak1, Sebastian Demkowicz1, Janusz Rachon1

  • 1Department of Organic Chemistry, Faculty of Chemistry, Gdansk University of Technology, Narutowicza 11/12, 80-233, Gdansk, Poland.

European journal of medicinal chemistry
|April 17, 2025
PubMed
概括

新型类固醇硫酶 (STS) 抑制剂被合成和测试. 化合物54E在酶和细胞分析中显示出高活性,具有临床前开发的潜力.

关键词:
癌症 癌症 癌症 癌症分子对接是分子对接.STS 抑制剂的使用.类固醇硫酸酶是一种类固醇.这种药物是三醇.

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