Factors Affecting Dissolution: Drug Permeability, Stability and Stereochemistry
Tagging and Fusion Proteins
Prodrugs
Olefin Metathesis Polymerization: Acyclic Diene Metathesis (ADMET)
Phosphoinositides and PIPs
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Dmitri Simberg1,2, Yechezkel Barenholz3, Steve R Roffler4,5
1Department of Pharmaceutical Sciences, The Skaggs School of Pharmacy and Pharmaceutical Sciences and Colorado Center for Nanomedicine and Nanosafety, University of Colorado Anschutz Medical Campus, Aurora, CO, USA.
聚乙烯甘醇 (PEG) 化增强了药物输送,但新出现的抗PEG抗体引发了安全问题. 需要进一步的研究,以了解免疫反应,并探索PEG替代品的未来药物.
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