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Updated: May 12, 2025

Preparation of Contiguous Bisaziridines for Regioselective Ring-Opening Reactions
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区域选择性,易斯酸催化环开放的2,3-阿齐里迪尔酒精与亚醇

Benjamin Zheng1, Mark S Taylor1

  • 1Department of Chemistry, University of Toronto, Toronto, Ontario M5S 3H6, Canada.

The Journal of organic chemistry
|April 25, 2025
PubMed
概括

研究人员使用阿醇核友来开发了N-硫尼尔保护的亚齐里基醇的区域选择性环开反应. 这种方法实现了高的C3选择性和N选择性,为复杂分子提供了一条新的合成路线.

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