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Updated: May 10, 2025

Functionalized Spirocyclic Heterocycle Synthesis and Cytotoxicity Assay
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在第1位和第10位中修改的新时代蛋白A类似物合成和生物研究

Dilyana Dimitrova1, Veronica Nemska1, Ivan Iliev2

  • 1Biotechnology Department, University of Chemical Technology and Metallurgy, 8 Kliment Ohridski Blvd., 1797 Sofia, Bulgaria.

Pharmaceutics
|April 26, 2025
PubMed
概括

修改的抗微生物 (AMP) 显示出对抗耐药性感染的承诺. 与Tyr或化Phe替代品类似的Temporin A显示出强大的抗菌和抗增殖活性,具有低毒性.

关键词:
一个临时的A.抗微生物活性的抗微生物活性.抗微生物类的抗微生物.它们具有抗增殖活性.细胞毒性 细胞毒性化氨基酸是一种化氨基酸.水溶性稳定性 水溶性稳定性摄影毒性 摄影毒性

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