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Updated: May 9, 2025

Preparation and Evaluation of 99mTc-labeled Tridentate Chelates for Pre-targeting Using Bioorthogonal Chemistry
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Preparation and Evaluation of 99mTc-labeled Tridentate Chelates for Pre-targeting Using Bioorthogonal Chemistry

Published on: February 4, 2017

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在线链和分支链结构之间比较碳酸盐无水酶-IX向的三功能放射性连接体

Kazuma Nakashima1, Takayoshi Ichinose1, Hiroyuki Watanabe1

  • 1Department of Patho-Functional Bioanalysis, Graduate School of Pharmaceutical Sciences, Kyoto University, Kyoto, Japan.

Frontiers in nuclear medicine
|May 1, 2025
PubMed
概括

与线性链版本相比,一个分支链放射性连接体 (In-DOTAGA-ALB-IS) 证明了优越的瘤向和减少脏吸收. 这表明分支设计可以提高CA-IX向放射性连体的有效性.

关键词:
CA-IX 是一个CA-IX.多塔是什么意思?多塔是什么意思?专蛋白绑定剂 专蛋白绑定剂有分支链的排列方式.在imidazothiadiazole硫胺中使用.线性链条的排列方式

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