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Updated: May 9, 2025

Preparation of Enantiopure Non-Activated Aziridines and Synthesis of Biemamide B, D, and epiallo-Isomuscarine
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切换酸酶与酶选择性水合活性,以有效合成基拉尔2,2-二甲基cyclopropanecarboxamide

Xiao-Ling Tang1,2, Xu-Gang Zhang1,2, Ye-Tao Zhang1,2

  • 1Key Laboratory of Bioorganic Synthesis of Zhejiang Province, College of Biotechnology and Bioengineering, Zhejiang University of Technology, Hangzhou, People's Republic of China.

Biotechnology and bioengineering
|May 1, 2025
PubMed
概括

研究人员设计了一种亚酶酶,以产生性2,2-二甲基cyclopropanecarboxamides,关键的制药中间体. 这种新的方法显著提高了胺合成效率和酶选择性,克服了以前的局限性.

关键词:
这是一种二二二二二二甲基cyclopropanecarboxamide.它们具有enantioselectivity的作用.补水活动的水合活性.亚酸酶的使用方法反应特异性的反应特异性.

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