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Updated: May 23, 2025

Establishing Dual Resistance to EGFR-TKI and MET-TKI in Lung Adenocarcinoma Cells In Vitro with a 2-step Dose-escalation Procedure
09:38

Establishing Dual Resistance to EGFR-TKI and MET-TKI in Lung Adenocarcinoma Cells In Vitro with a 2-step Dose-escalation Procedure

Published on: August 11, 2017

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开发新的抗癌类硫胺作为EGFR/碳酸无水酶双抑制剂的新型抗癌药物

Ibrahim H Eissa1, Hazem Elkady1, Walid E Elgammal2

  • 1Pharmaceutical Medicinal Chemistry & Drug Design Department, Faculty of Pharmacy (Boys), Al-Azhar University, Cairo, Egypt.

Future medicinal chemistry
|May 8, 2025
PubMed
概括

新的硫胺衍生物显示出作为表皮生长因子受体 (EGFR) 和碳酸酶IX (CA-IX) 的双重抑制剂的潜力,用于选择性抗癌疗法.

关键词:
这是一种抗癌药物.细胞亡,计算研究研究.药物设计 药物设计双 EGFR - 碳酸无水酶抑制剂亚二 - 硫胺胺 硫胺 硫胺 硫胺

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Development and Maintenance of a Preclinical Patient Derived Tumor Xenograft Model for the Investigation of Novel Anti-Cancer Therapies09:29

Development and Maintenance of a Preclinical Patient Derived Tumor Xenograft Model for the Investigation of Novel Anti-Cancer Therapies

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