新瑞衍生物的药理动力学预测和细胞毒性

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Michele Goulart Dos Santos1, Marie Demonceaux2, Lucia Emanueli Schimith3

  • 1Programa de Pós-Graduação em Ciências Fisiológicas, Instituto de Ciências Biológicas, Universidade Federal do Rio Grande, Rio Grande, Rio Grande do Sul, Brazil.

Chemistry & biodiversity
|May 9, 2025
PubMed
概括

昆素 (QUE) 的酶性糖基化产生了新的α-糖基化衍生物. 这些衍生物显示出改善的药理动力学,并且与原始奎尔塞丁及其β-葡萄糖化形式不同,无毒.

关键词:
在ADME的分析中,ADME分析了细胞毒性 细胞毒性这种类型的黄类药物是flavonoid.物理化学特性 物理化学特性转葡萄糖化转糖化

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