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Updated: May 12, 2025

A Method for Screening and Validation of Resistant Mutations Against Kinase Inhibitors
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小分子激酶抑制剂在癌症治疗中的心脏毒性

Shuangli Zhu1, Kai Fu1, Sijia Li1

  • 1State Key Laboratory of Oncology in South China, Collaborative Innovation Center for Cancer Medicine, Guangdong Esophageal Cancer Institute, Guangdong Provincial Clinical Research Center for Cancer, Sun Yat-Sen University Cancer Center, Guangzhou, 510060, Guangdong, People's Republic of China.

Experimental hematology & oncology
|May 9, 2025
PubMed
概括

小分子激酶抑制剂 (SMKI) 是有效的癌症治疗方法,但可能导致心脏毒性. 本综述总结了SMKI心脏毒性机制和预防和设计更安全药物的策略.

关键词:
癌症 癌症 癌症 癌症心脏有毒性 - 心脏有毒性小分子激酶抑制剂 小分子激酶抑制剂

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