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Updated: May 15, 2025

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作为抗癌剂的纳夫托金盐的设计,合成和生物评估

Yao Cheng1, Tsz Tin Yu1, Ellen M Olzomer2

  • 1School of Chemistry, University of New South Wales, Sydney, NSW 2052, Australia.

Molecules (Basel, Switzerland)
|May 14, 2025
PubMed
概括

研究人员开发了基于BH10的新盐化合物,以准癌症中的华堡效应. 化合物7b通过与Keap1相互作用,显示出显著的抗癌活性和选择性,提供了一个有前途的治疗策略.

关键词:
这是一种抗癌药物.葡萄糖溶解是什么纳夫托伊米达 (naphthoimidazole) 是一种天然的药物.选择性的选择性

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