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Updated: May 17, 2025

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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Published on: February 20, 2018

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比较CB1和CB2受体之间的激素活性与正位突变之间的激素活性

Christina A Brust1,2, Matthew A Swanson1,2, Christos Iliopoulos Tsoutsouvas3

  • 1The Herbert Wertheim UF Scripps Institute for Biomedical Innovation and Technology, Department of Molecular Medicine, Jupiter, FL 33458, USA.

Receptors (Basel, Switzerland)
|May 16, 2025
PubMed
概括

研究大麻素受体 (CB1和CB2) 发现,突变的特定残留物会以不同的方式影响它们的功能. 这项研究有助于通过了解受体亚型敏感性来开发治疗疼痛和炎症的选择性药物.

关键词:
AM1203333 是一个很好的公司.在CP55,94040中使用.G蛋白结合受体的受体是G蛋白结合受体的受体.大麻素是一种大麻素.在内部化,内化.

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