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Updated: May 20, 2025

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一种酸降低异构酶抑制剂,具有抗结核和除草剂活性

Luke William Guddat1, Xin Lin2, Julia L Kurz3

  • 1The University if Queensland, School of Chemistry and Molecular Biosciences, Cooper Rd, 4072, Brisbane, AUSTRALIA.

Chemistry (Weinheim an der Bergstrasse, Germany)
|May 19, 2025
PubMed
概括

针对酸还原异构酶 (KARI) 的新生物杀伤剂显示出有前途. 化合物1f抑制了Mycobacterium tuberculosis KARI,显示出开发针对植物和微生物病原体的有效生物制剂的潜力.

关键词:
药物发现 药物发现凯酸还原化异构酶晶体结构 晶体结构除草剂的发现除草剂的发现抑制剂抑制剂的使用

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