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Updated: Sep 17, 2025

Preparation of Enantiopure Non-Activated Aziridines and Synthesis of Biemamide B, D, and epiallo-Isomuscarine
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作为潜在的胆酶抑制剂的奇拉尔人体胺基:合成,生物活性评估和分子建模

Turgay Tunç1, Namık Kılınç2, Nadir Demirel3

  • 1Department of Chemistry Engineering and Process, Faculty of Engineering, University of Kırşehir Ahi Evran, Kırşehir, Türkiye.

Chemistry & biodiversity
|July 2, 2025
PubMed
概括

新型性人类氨基胺显示出对乙胆酶 (AChE) 和丁胆酶 (BChE) 的强烈抑制,这是阿尔茨海默病 (AD) 的关键标. 观察到对抗选择性抑制,特定的异构体显示出对 AChE 和 BChE 的优越疗效.

关键词:
乙烯基胆化酶的使用甲基胆化酶 (butyrylcholinesterase) 是一种基胆化酶.合性人类胺.抑制抑制抑制的抑制作用分子对接的分子对接.

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