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Updated: Sep 17, 2025

Parallel Interrogation of β-Arrestin2 Recruitment for Ligand Screening on a GPCR-Wide Scale using PRESTO-Tango Assay
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在GPCR药理学中的可光切换的全和双联体

Silvia Mori1, Damiano Arella1, Michael Decker1

  • 1Julius Maximilian University Würzburg (JMU), Institute for Pharmacy and Food Chemistry, Pharmaceutical and Medicinal Chemistry, 97074 Würzburg, Germany.

Trends in pharmacological sciences
|July 2, 2025
PubMed
概括

研究人员正在开发新的可光开关联体,以精确控制使用光的G蛋白合受体 (GPCRs). 这些全和双化合物提供了增强的选择性和对受体功能的精细控制,推进了光药学.

关键词:
BQCA BQCA 这是一个很好的例子.亚烯是什么 亚烯是什么 阿烯是什么药物设计 药物设计葡萄糖酸盐受体的受体摄影药理学 摄影药理学接收器动态 接收器动态

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