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Updated: Sep 16, 2025

Solid-phase Synthesis of [4.4] Spirocyclic Oximes
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Published on: February 6, 2019

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无痕基集团指导策略:聚环类化物支架的模块化合成

Qing Li1, Yuting Zhao2, Xinyu Zhu1

  • 1Department of Medicinal Chemistry, China Pharmaceutical University, 211198 Nanjing, China.

Organic letters
|July 9, 2025
PubMed
概括

这项研究引入了一种新的-曼尼克/乳酸化/酸消除级联. 这种方法有效地构建复杂的piperidone和isoquinolone化物支架,使用化作为无痕指导组.

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