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Updated: Sep 15, 2025

Preparation of Enantiopure Non-Activated Aziridines and Synthesis of Biemamide B, D, and epiallo-Isomuscarine
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Published on: June 13, 2022

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通过宏循环化/跨环 pyran 循环化策略的 (-) - Enigmazole A 的总合成:应用于结构-活动关系调查的应用

Kyoya Ohyama1, Taisei Masuda1, Keita Sakamoto1

  • 1Department of Applied Chemistry, Faculty of Science and Engineering, Chuo University, 1-13-27 Kasuga, Bunkyo-ku, Tokyo 112-8551, Japan.

The Journal of organic chemistry
|July 15, 2025
PubMed
概括

通过一种新的宏循环化策略,实现了 (-) - 益格马 A 的 18 步总合成. 这种方法构建了麦克罗拉克骨架,并使得用于结构-活性关系研究的类似物能够产生.

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