核性α-和β-添加物使结合胺酸的氧-中性亚齐化成为可能

Rui Wang1, Quanbin Jiang1, Long Jiang2

  • 1School of Chemistry, Sun Yat-sen University, Guangzhou 510006, P. R. China.

概括

这项研究引入了一种使用非受保护的初级氨基和内部氧化剂的新方法,克服了直接氧化的挑战. 这种方法可以从简单的前体中合成复杂的阿齐里丁和N-阿里尔阿齐里丁.

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