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Updated: Sep 15, 2025

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准电压通的质子通道HV1:优化了具有抗癌潜力的5--2-氨基胺醇

Martina Piga1, Geraldo Jorge Domingos2, Adam Feher2

  • 1Faculty of Pharmacy, University of Ljubljana, Aškerčeva cesta 7, Ljubljana, 1000, Slovenia.

European journal of medicinal chemistry
|July 15, 2025
PubMed
概括

新的电压关闭质子通道 (HV1) 抑制剂在治疗癌症和神经炎症等疾病方面表现有前途. 优化的化合物表现出强大的抗增殖作用,特别是在具有高HV1表达的细胞中,推进治疗策略.

关键词:
5 - -2-氨基胺基胺醇的使用.这是一种抗癌药物.H (((V) 1 一个抑制剂的抑制剂电压通的质子通道.

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