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Updated: Sep 13, 2025

Optimization of the Ugi Reaction Using Parallel Synthesis and Automated Liquid Handling
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使用Umpolung胺合成合成的费格利米的总合成

Preston C Gourville1, Jade A Bing1, Rashanique D Quarels1

  • 1Department of Chemistry, Institute of Chemical Biology, Vanderbilt University, Nashville, TN, USA.

Angewandte Chemie (International ed. in English)
|July 27, 2025
PubMed
概括

这项研究引入了胺合成 (UmAS) 用于制备,简化了复杂的步骤,并使非正规残留物的反选择性合成成为更绿色的药物发现.

关键词:
抗病毒药物是一种抗病毒药.乙选择性胺基合成费格利米辛是一种药物.自然产品的合成方法乌姆波隆胺合成方法

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