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Updated: Sep 13, 2025

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硫胺组修改对塞莱科西布的影响:矩阵金属蛋白酶交互性UTX-121衍生物的分子特征

Kazuto Ohkura1, Atsushi Tabata2, Yoshihiro Uto2

  • 1Graduate School of Pharmaceutical Sciences, Suzuka University of Medical Science, Suzuka, Japan; kohkura@suzuka-u.ac.jp.

Anticancer research
|August 1, 2025
PubMed
概括

一种新的UTX-121衍生物a2通过强烈抑制矩阵甲蛋白酶-2 (MMP-2) 来证明增强抗瘤活性. 这种衍生品对开发针对MMP-2的新抗癌疗法充满希望.

关键词:
在MMP中,MMP是MMP.分子设计分子设计.在UTX-12121中使用.

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