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Updated: Sep 12, 2025

Regioselective O-Glycosylation of Nucleosides via the Temporary 2',3'-Diol Protection by a Boronic Ester for the Synthesis of Disaccharide Nucleosides
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Regioselective O-Glycosylation of Nucleosides via the Temporary 2',3'-Diol Protection by a Boronic Ester for the Synthesis of Disaccharide Nucleosides

Published on: July 26, 2018

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乌拉衍生物/乌尔索酸混合物 - 作为抗癌剂的天然衍生物化合物

Olga Michalak1, Marcin Cybulski2, Marek Kubiszewski3

  • 1Chemistry Section; Pharmacy, Cosmetic Chemistry and Biotechnology Research Group, Łukasiewicz Research Network-Industrial Chemistry Institute, 8 Rydygiera Str, Warsaw, 01-793, Poland. olga.michalak@ichp.lukasiewicz.gov.pl.

Scientific reports
|August 6, 2025
PubMed
概括

新的 uracil-ursolic 酸混合体对乳腺癌细胞系表现出强大的抗癌活性. 化合物6a有效地降低了细胞活力和抑制了Akt激酶,显示出作为新型细胞毒性剂的潜力.

关键词:
ADME ADME ADME ADME ADME ADME ADME ADME ADME ADME ADME ADME ADME ADME ADME ADME ADME ADME ADME ADME ADME ADME ADME ADME ADME ADME ADME ADME ADME ADME ADME ADME ADME ADME ADME ADME ADME乳腺癌 乳腺癌 乳腺癌细胞毒性活动的细胞毒性.分子对接是分子对接.乌拉衍生物的衍生品乌尔索利酸是什么 乌尔索利酸是什么

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Uracil-DNA Glycosylase Assay by Matrix-assisted Laser Desorption/Ionization Time-of-flight Mass Spectrometry Analysis12:19

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