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Updated: Sep 11, 2025

Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
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Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission

Published on: August 16, 2018

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检查由内分泌大麻素诱导的格拉米西丁电流的变化.

Sultan Mayar1, Audrey Cyr-Athis1, Nazzareno D'Avanzo1

  • 1Université de Montréal, Département de pharmacologie et physiologie, Montréal, Québec, Canada.

PloS one
|August 18, 2025
PubMed
概括

内分类固醇,影响神经系统的关键脂质,可以通过改变膜性质来改变离子通道功能. 特定的2-单糖醇 (2-MG) 显示了它们的结构和对格拉米西丁电流的影响之间的相关性.

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