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Updated: Sep 10, 2025

A Method for Screening and Validation of Resistant Mutations Against Kinase Inhibitors
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使用BTK抑制剂TL-895的药物相互作用负担

Jack C Stromatt1, Eman A Ahmed1, Thomas Drabison1

  • 1The Ohio State University, Columbus, Ohio, United States.

Cancer research communications
|August 22, 2025
PubMed
概括

这是一种双BTK/ BMX抑制剂,具有强烈的BMX抑制作用. 它是OATP1B1和CYP3A4的基质,但不太可能引起药物相互作用,确保在组合治疗中使用更安全.

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