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Updated: Sep 10, 2025

A Simple Bioassay for the Evaluation of Vascular Endothelial Growth Factors
09:04

A Simple Bioassay for the Evaluation of Vascular Endothelial Growth Factors

Published on: March 15, 2016

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作为VEGFR-2抑制剂的1,3,4-提亚衍生物及其癌症治疗的分子洞察力

Pragya Gawande1, Balaji Wamanrao Matore1, Anjali Murmu1

  • 1Laboratory of Drug Discovery and Ecotoxicology, Department of Pharmacy, Guru Ghasidas Vishwavidyalaya (A Central University), Bilaspur, Chhattisgarh, India.

Chemistry & biodiversity
|August 26, 2025
PubMed
概括

作为针对血管内皮生长因子受体-2 (VEGFR-2) 的新型抑制剂,1,3,4- 亚醇衍生物在癌症治疗中具有前景. 与现有治疗方法相比,这些化合物具有提高选择性和降低毒性的潜力.

关键词:
一,三,四-亚血管新生癌症结构活动关系 (SAR) 和机制血管内皮生长因子受体-2 (VEGFR-2) 抑制剂

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