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Updated: Sep 10, 2025

Measuring G-protein-coupled Receptor Signaling via Radio-labeled GTP Binding
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通过偏差和GRK亚型分辨出AT1R的酸化模式

Zisu Zhang1, Chuyi Liu2, Jinda Gong1

  • 1The Second Affiliated Hospital of Zhejiang University School of Medicine, Research Center for Clinical Pharmacy, Key Laboratory of Neuropharmacology and Translational Medicine of Zhejiang Province, State Key Laboratory of Advanced Drug Delivery and Release Systems, Institute of Pharmacology and Toxicology, College of Pharmaceutical Sciences, Zhejiang University, Hangzhou 310058, China.

International journal of molecular sciences
|August 28, 2025
PubMed
概括

不同的激动剂和GPCR激酶 (GRKs) 产生独特的血管激素II类型1受体 (AT1R) 酸化模式,影响β- 逮捕素的招募. 了解这些条形码有助于AT1R治疗的发展.

关键词:
在AT1R土耳其有偏见的连接体化维生素B的含量

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