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Updated: Sep 9, 2025

Author Spotlight: Developing Acetyl-Click Assay for HAT1 Inhibitor Screening
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在确定下一代乙胆酶抑制剂方面的计算见解和实验突破

Devaraj Hanumanthappa1, Bandral Sunil Kumar1, Sandra Ross Olakkengil Shajan2

  • 1Department of Pharmaceutical Chemistry, Faculty of Pharmacy, M.S. Ramaiah University of Applied Sciences, Bengaluru, 560054, Karnataka, India.

Scientific reports
|August 29, 2025
PubMed
概括

这项研究将莱特作为潜在的阿尔茨海默氏症治疗方法,将其制成固体脂质纳米颗粒 (L-SLN). 在阿尔茨海默氏症小鼠模型中,L-SLN表现出显著的神经保护作用,突显了它们的治疗潜力.

关键词:
乙胆酶阿尔茨海默病药物重新使用莱特固体脂质纳米粒子

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