Ligand Binding and Linkage
Conserved Binding Sites
Cooperative Binding of Transcription Regulators
Ligand Binding Sites
The Equilibrium Binding Constant and Binding Strength
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Daniel R Fox1, Cyntia Taveneau2, Janik Clement3
1Department of Biochemistry and Pharmacology, Bio21 Molecular Science and Biotechnology Institute, The University of Melbourne, Parkville, VIC 3010, Australia; Department of Microbiology, Biomedicine Discovery Institute, Monash University, Clayton, VIC 3800, Australia; Centre for Electron Microscopy of Membrane Proteins, Monash Institute of Pharmacological Sciences, Parkville, VIC 3052, Australia; AI Protein Design Program, Biomedicine Discovery Institute, Monash University, Clayton, VIC, 3800, Australia.
结构生物学中的人工智能使得新蛋白质的设计成为可能. 机器学习加速了对挑战性目标的高亲和度结合剂的开发,
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