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Updated: Sep 9, 2025

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来自TLQP-21的新型补充3a受体激活剂和对抗剂

Pedro Rodriguez1, Jean Pierre Pallais1, Rongjun He2

  • 1Department of Integrative Biology and Physiology, University of Minnesota, Minneapolis, Minnesota 55455, United States.

Journal of medicinal chemistry
|September 3, 2025
PubMed
概括

研究人员通过创建新的类型来优化补充3a受体 (C3aR). 这些修改增强了C3aR信号的选择性和效力,为炎症,代谢和神经疾病提供了新的治疗途径.

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