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Updated: Sep 9, 2025

Preparation of N-2-alkoxyvinylsulfonamides from N-tosyl-1,2,3-triazoles and Subsequent Conversion to Substituted Phthalans and Phenethylamines
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Preparation of N-2-alkoxyvinylsulfonamides from N-tosyl-1,2,3-triazoles and Subsequent Conversion to Substituted Phthalans and Phenethylamines

Published on: January 3, 2018

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探索对Sydnones的激进添加:一个通往 perfluoroalkyl-substituted pyrazoles的通道

Zakhar M Rubanov1, Denis S Koltun1, Vitalij V Levin1

  • 1N. D. Zelinsky Institute of Organic Chemistry, Leninsky Prospekt 47, Moscow 119991, Russian Federation.

Organic letters
|September 4, 2025
PubMed
概括

这项研究引入了一种直接添加到sydnones的新方法,从而产生化化合物. 这些化合物随后用于合成药用化学的重要 perfluoroalkylated pyrazole.

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