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Updated: Sep 9, 2025

An Efficient Method for the Synthesis of Peptoids with Mixed Lysine-type/Arginine-type Monomers and Evaluation of Their Anti-leishmanial Activity
12:02

An Efficient Method for the Synthesis of Peptoids with Mixed Lysine-type/Arginine-type Monomers and Evaluation of Their Anti-leishmanial Activity

Published on: November 2, 2016

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含尿素的衍生物的合成及其作为潜在的抗甲基耐药性Aureus葡萄球菌剂的应用

Jorge A González-Cruz1, Gerardo González-Gallardo1, J Ricardo Pérez-Velázquez2

  • 1Departamento de Química Orgánica, Instituto de Química, Universidad Nacional Autónoma de México (UNAM), Ciudad de México, 04510, México.

ChemMedChem
|September 5, 2025
PubMed
概括

新的含尿素的胺基对抗甲素耐药黄金葡萄球菌 (MRSA) 有潜力. 这些化合物被设计为已知的抑制剂的生物分离物,有效地抑制了细菌的生长,表明FabI是潜在的分子标.

关键词:
制造蛋白抑制剂抗微生物耐药性甲素耐药的金色葡萄球菌分子对接尿素衍生物

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