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Updated: Jan 18, 2026

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罗沙沙斯塔特激活甲状腺激素受体α和β在临床相关度

Koji Morita1, Toru Iigo1, Kaho Jimbo1

  • 1Division of Endocrinology and Metabolism, Department of Internal Medicine, Teikyo University School of Medicine, Tokyo, JPN.

Cureus
|September 12, 2025
PubMed
概括

用于治疗脏贫血的罗沙杜沙特可能会激活甲状腺激素受体 (TRα和TRβ). 这项研究发现,roxadustat在基于细胞的测定中激活了这些受体,这表明在临床剂量下具有潜在的甲状腺学活性.

关键词:
缺氧诱导因子-普罗利尔氧酶抑制剂光酶测定试验罗克萨斯达斯塔特的情况甲状腺激素受体 甲状腺激素受体甲状腺神经活动的活性.

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