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Updated: Jan 17, 2026

Quantitative Structure-Activity Relationship, Activity Prediction, and Molecular Dynamics of Non-nucleotide Reverse Transcriptase Inhibitors
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提亚-碳胺衍生物作为具有药物类似性能的强有力的抗氧化剂:体外,分子对接和DFT研究

Mohammed Hawash1, Dina Ghannam1, Leen Dawoud1

  • 1Department of Pharmaceutical Chemistry and Technology, Faculty of Pharmacy, An-Najah National University, Nablus, Palestine.

PloS one
|September 19, 2025
PubMed
概括

新合成的 thiazole-carboxamide 衍生物显示出强大的抗氧化活性,超过了 Trolox. 虽然这些化合物具有较弱的抗糖尿病潜力,但它们在口服时具有很好的药物相似性,为进一步的治疗研究铺平了道路.

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