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Updated: Jan 14, 2026

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一些7-基氨酸化合物的对凝血因子Xa,尿素酶和抗糖尿病酶的影响

Furkan Meletli1, Ayşe Ogan1, Refiye Yanardag2

  • 1Department of Chemistry, Faculty of Science, Marmara University, Istanbul, Turkey.

Bioorganic chemistry
|October 17, 2025
PubMed
概括

合成了六种新的氨酸-甲二混合物,并对酶抑制进行了测试. 化合物K3和K8对XA因子和α-葡萄糖酶分别表现出强烈的活性,这表明了潜在的治疗应用.

关键词:
库马林 - 甲二烯混合物在 FXaXa FXa分子对接是分子对接.在Urease中使用Urease.α-氨基酶的使用.α-葡萄糖化酶的使用.

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