抑制HSP90 破坏单细胞细胞中27-基胆固醇诱导的炎症信号

Jaesung Kim1, Munju Kwon2, Dongha Park1

  • 1Department of Pharmacology, School of Medicine, Pusan National University, Yangsan 50612, Republic of Korea.

概括

用ganetespib抑制热冲击蛋白90 (HSP90) 降低了单细胞细胞中胆固醇代谢物27-基胆固醇 (27OHChol) 诱导的炎症. 这种有针对性的方法抑制了关键的炎症途径,为代谢炎症提供了潜在的治疗益处.