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Updated: Jan 13, 2026

Development of Inhibitors of Protein-protein Interactions through REPLACE: Application to the Design and Development Non-ATP Competitive CDK Inhibitors
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针对选择性抑制CLK3激酶的研究

Vinay Kumar Singh1,2, Frédéric Justaud1, Dabbugoddu Brahmaiah3

  • 1Univ Rennes, CNRS, ISCR (Institut des Sciences Chimiques de Rennes), UMR 6226, F-35000 Rennes, France.

Beilstein journal of organic chemistry
|October 29, 2025
PubMed
概括

科学家们开发了VS-77,这是一个强大的抑制剂,向CLK3激酶,对于mRNA拼接至关重要. 这一发现促进了对CLK3的理解.

关键词:
在 CLK3 中,癌症 癌症 癌症 癌症 癌症激酶激酶是一种激素.分子建模分子建模纳胺是一种胺.有三醇的三醇.

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