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Updated: Jan 12, 2026

High Content Screening Analysis to Evaluate the Toxicological Effects of Harmful and Potentially Harmful Constituents HPHC
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在hCB1上流行的合成大麻素代谢物的结构-活性关系 in vitro 和 in silico动态

Anna Åstrand1, Emiliano Laudadio2, Prince S Gameli3

  • 1Division of Clinical Chemistry and Pharmacology, Department of Biomedical and Clinical Sciences, Faculty of Medicine and Health Sciences, Linköping University, SE 581 85 Linköping, Sweden. anna.astrand@liu.se.

Acta pharmacologica Sinica
|November 3, 2025
PubMed
概括

合成大麻素代谢物被测试在人类大麻素受体1 (hCB) 的活性. 许多代谢物保留了显著的疗效,其中4-基烯衍生物显示出高强度,这表明它们有助于合成大麻素效应.

关键词:
活性代谢物的活性代谢物.在形对接和分子动力学中.药理动力学是药理动力学的一个方面.结构-活动关系关系.合成大麻素受体激活剂 合成大麻素受体激活剂

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